Proteins
This section lists all Axon Ligands™ that interact with proteins that do not show enzymatic activity or transduce signals by any signaling pathway mechanism. Among the pharmacological tools listed here are ligands that interact with transporters of any kind, proteins that affect intra- and/or extracellular structures, and proteins that assist enzymes without showing catalytic activity by itself.
| Axon ID | Name | Description | From price | |
|---|---|---|---|---|
| 3755 | (+)-Abscisic acid | LANCL2 ligand | €90.00 | |
| 1989 | (+)-JQ1 |
Potent and selective BET bromodomain inhibitor |
€60.00 | |
| 3822 | (+)-JQ1 carboxylic acid | (+)-JQ1 derivative; PROTAC precursor | €110.00 | |
| 3873 | (-)-JQ-1 | Inactive enantiomer of (+)-JQ1 | €120.00 | |
| 3777 | (R)-AS-1 | First-in-class highly selective and orally bioavailable PAM of EAAT2 | €145.00 | |
| 2830 | (R)-CE3F4 | Potent inhibitor of EPAC1 | €120.00 | |
| 3928 | (R)-SKBG-1 | Covalent RNA-binding protein NONO ligand | €160.00 | |
| 4192 | (S)-BI 2536 | Dual PLK1/BRD4 bromodomain inhibitor | €170.00 | |
| 3929 | (S)-SKBG-1 | Inactive enantiomer of (R)-SKBG-1 | €150.00 | |
| 3617 | 1R,3R-RSL3 (negative control) | Negative control of 1S,3R-RSL3 as GPX4 inhibitor | €90.00 | |
| 3957 | A-1155463 dihydrochloride | BH3 mimetic Ligand of BCL protein BCL-XL | Inquire | |
| 4008 | A-1210477 | Potent and selective inhibitor of MCL-1 | Inquire | |
| 3972 | A-1331852 | BH3 mimetic Ligand of BCL protein BCL-XL | €120.00 | |
| 3696 | ABBV-075 | Highly potent and orally bioavailable BET bromodomain (BRD) inhibitor | €110.00 | |
| 4263 | ABBV-467 | Potent and selective MCL-1 inhibitor | Recently added | Inquire |
| 3956 | ABBV-744 | First-in-class highly BDII (Bromodomain II)-selective BET bromodomain inhibitor | Inquire | |
| 3564 | ABCA1 inducer compound G | ABCA1 inducer targeting OSBPL7 | €150.00 | |
| 3631 | ABR-238901 | Potent S100A8/A9 blocker | €170.00 | |
| 2141 | ABT 199 | Potent, orally bioavailable BCL-2-selective inhibitor | €70.00 | |
| 3821 | ABT-263 | Potent, selective and orally bioavailable inhibitor of B-cell lymphoma-2 (BCL-2) family proteins | Inquire | |
| 2552 | Adjudin | Non-hormonal male contraceptive with anti-proliferative activity | €125.00 | |
| 3687 | ADU-S100 | Cyclic dinucleotide (CDN) agonist (activator) of Stimulator of Interferon Genes (STING) | Inquire | |
| 4175 | AJ2-30 | First-in-class SLC15A4 inhibitor | €110.00 | |
| 1238 | ALX 5407 hydrochloride | GlyT-1 inhibitor | €140.00 | |
| 3686 | AMG-176 | Potent and selective Mcl-1 inhibitor | €490.00 | |
| 1333 | Amoxapine | Tricyclic antidepressant; Potent reuptake inhibitor of norepinephrine (NRI) | €50.00 | |
| 3433 | ARB-272572 | Potent, cellular active PD-L1 inhibitor | €150.00 | |
| 2941 | ARN 272 | Selective inhibitor of FAAH-like anandamide transporter (FLAT) | €90.00 | |
| 3944 | ARV-825 | Potent and selective protein BRD4 degrader | Inquire | |
| 1297 | Atomoxetine hydrochloride | NRI inhibitor | €95.00 | |