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Momelotinib hydrochloride - CYT387 hydrochloride

Based on 158 reference(s) in Google Scholar 8 10 158

Axon 4124

CAS [1841094-16-3]

MF C23H22N6O2.HCl
MW 450.92

  • Purity: 98%
  • Soluble in DMSO

Momelotinib hydrochloride

Description

Selective and ATP-competitive Janus Kinase JAK1/JAK2 inhibitor, with IC50 to be 11 and 18 nM for JAK1 and JAK2 respectively and far less activity against other kinases, including JAK3 (IC50=155 nM). The free base, Momelotinib (Axon 1681) is also available.

Keywords: Momelotinib hydrochloride | Supplier | JAK1/2 inhibitor | CYT387 hydrochloride | CYT-387 | CYT 387 | CAS [1841094-16-3] | [1056634-68-4] | [1380317-28-1] | [1841094-17-4] | JAK-STAT Pathway | JAK | Inhibitor | Enzymes

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Size Unit Price Stock
10 mg €120.00 In Stock
50 mg €360.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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