CEP-33779

Based on 16 reference(s) in Google Scholar 8 10 16

Axon 3671

CAS [1257704-57-6]

MF C24H26N6O2S
MW 462.57

CEP-33779

Description

CEP-33779 is a potent, selective and orally bioavailable JAK2 inhibitor with an IC50 value of 1.8 nM.

Cell Signaling & Oncology Pain & Inflammation JAK-STAT EC 2.7.10.2 JAK

Potent, selective and orally bioavailable JAK2 inhibitor

N-(3-(4-Methylpiperazin-1-yl)phenyl)-8-(4-(methylsulfonyl)phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine

[1257704-57-6]

Order

Size	Unit Price	Stock
5 mg	€95.00	In Stock
25 mg	€290.00	In Stock

Need more? Bulk Inquiry

Axon ID	Name	Description
1378	AG 490	JAK2 inhibitor	€65.00
1588	TG 101348	JAK2 inhibitor	€80.00
1598	Ruxolitinib	JAK1 and JAK2 inhibitor	€65.00
1681	Momelotinib	JAK1 and JAK2 inhibitor	€80.00
1778	AZ 960	JAK2 inhibitor	€95.00
1843	JAK2 inhibitor 13	JAK2 inhibitor	€110.00
1955	Baricitinib	Inhibitor of JAK1 and JAK2	€70.00
2219	AT 9283	Multitargeted kinase inhibitor (Aurora A/B, JAK2/3, and BCR-Abl)	€85.00
2231	XL 019	JAK2 inhibitor	€100.00
2316	WP 1066	Potent JAK2 and STAT3 inhibitor and downregulator of antiapoptotic proteins	€95.00
2554	LY 2784544	Potent, selective and ATP-competitive inhibitor of mutated janus kinase 2 (JAK2V617F)	€95.00
2658	MPT0B098	Microtubule inhibitor that suppresses JAK2/STAT3 signaling	€105.00
2792	NVP-BSK805	Potent, selective and orally bioavailable JAK2 inhibitor	€125.00
3813	BMS-911543	Potent, selective and orally active inhibitor of JAK2	Inquire
3855	AZD-4205	Selective and ATP-competitive inhibitor of JAK1	Inquire
3950	Peficitinib	Potent and orally bioavailable JAK inhibitor	€120.00
3997	ASN-002	Potent dual inhibitor of SYK and pan-JAK kinases	Inquire
4006	GLPG-0634	The first orally-available, selective inhibitor of JAK1	Inquire
4124	Momelotinib hydrochloride	JAK1 and JAK2 inhibitor	€120.00