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JAK2 inhibitor 13 - Sulfonamide 13

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1843

CAS [1110502-30-1]

MF C17H20N4O2S
MW 344.43

  • Purity: 99%
  • Soluble in DMSO

JAK2 inhibitor 13

Description

Potent and selective Janus Kinase 2 (JAK2) inhibitor; inhibits the activity of both the wild-type JAK2 and the V617F mutant (IC50 = 78 and 206 nM, respectively), with >35-fold selectivity versus JAK3 (IC50 = 2.93 µM)
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Size Unit Price Stock
5 mg €110.00 In Stock
25 mg €370.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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