CDK inhibitor CR8 - (R)-CR8

Based on 7 reference(s) in Google Scholar 8 10 7

Axon 3228

CAS [294646-77-8]

MF C24H29N7O
MW 431.53

  • Purity: 99%
  • Optical purity: 100% e.e.
  • Soluble in 0.1N HCl(aq) and DMSO
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CDK inhibitor CR8

Description

CDK inhibitor CR8 is a potent cyclin-dependent kinase (CDK) inhibitor with IC50 values of 0.09, 0.072, 0.041, 0.11, 1.10 and 0.18 μM for CDK1/cyclin B, CDK2/cyclin A, CDK2/cyclin E, CDK5/p25, CDK7/cyclin H and CDK9/cyclin T, respectively. Moreover, CDK inhibitor CR8 acts as a molecular glue degrader that depletes cyclin K.

KEYWORDS: CDK inhibitor CR8 | supplier | CDK inhibitor | (R)-CR8 | CDK inhibitor CR 8 | CDK inhibitor CR-8 | (R)-CR 8 | (R)-CR-8 | CAS [294646-77-8] | [1786438-30-9] | Cyclin Dependent (CDK) | CDK | Inhibitor | Enzymes

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5 mg €130.00 In Stock
25 mg €460.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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