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AR-42

Based on 47 reference(s) in Google Scholar 8 10 47

Axon 2394

CAS [935881-37-1]

MF C18H20N2O3
MW 312.36

  • Purity: 99%
  • Optical purity: optically pure
  • Soluble in DMSO

AR-42

Description

AR-42 is a novel HDAC inhibitor (IC50 value of 16 nM) with potent anticancer effects in pancreatic cancer cells at submicromolar concentrations by inducing cell cycle arrest, stimulating apoptosis, and regulating expression of several miRNAs. Also demonstrated anticancer activity in many other cancers, including acute myeloid leukemia, multiple myeloma, prostate cancer, ovarian cancer, human glioma cells, and bladder cancer.

KEYWORDS: AR-42 | supplier | HDAC inhibitor | AR 42 | AR42 | CAS [935881-37-1] | Histone | HDAC | Inhibitor | Enzymes

Order
Size Unit Price Stock
10 mg €125.00 In Stock
50 mg €450.00 In Stock
Special Offers
Size Unit Price Stock
2 x 10 mg €200.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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