CTEP - RO 4956371

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1972

CAS [871362-31-1]

MF C19H13ClF3N3O
MW 391.77

  • Purity: 99%
  • Soluble in DMSO

CTEP

Description

Potent, orally bioavailable, long lasting and selective mGluR5 allosteric antagonist or negative allosteric modulator; CTEP binds mGluR5 with low nanomolar affinity and shows >1000-fold selectivity against other targets, including all known mGlu receptorsCTEP has considerably improved properties over older mGluR5 antagonists such as MPEP (Axon 1222) and Fenobam (Axon 1345)

KEYWORDS: CTEP | supplier | NAM of mGluR5 | RO 4956371 | RO4956371 | CAS [871362-31-1] | Glutamate | mGluR5 | NAM | allosteric modulator | mpep | fenobam | long lasting

Order
Size Unit Price Stock
5 mg €120.00 In Stock
25 mg €420.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €180.00 In Stock
2 x 25 mg €640.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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