Your cart

There are no items in your shopping cart

AZD6244 - ARRY 142886 | Selumetinib

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1516

CAS [606143-52-6]

MF C17H15BrClFN4O3
MW 457.68

  • Purity: 99%
  • Soluble in DMSO

AZD6244

Description

An orally active, highly potent and selective inhibitor of MEK 1/2 that has shown tumor-suppressive activity in a wide range of preclinical models. IC50 value to be 14 nM against purified MEK1
Order
Size Unit Price Stock
5 mg €60.00 In Stock
25 mg €160.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €80.00 In Stock
2 x 25 mg €220.00 In Stock
Need more? Bulk Inquiry

Related Products

Axon ID Name Description From price
1122 SL 327 MEK1 and MEK2 inhibitor €80.00
1223 PD98059 MEK inhibitor €80.00
1357 SD 169 MAPK inhibitor (p38α specific) €60.00
1358 BIRB 796 MAPK inhibitor (p38 specific) €65.00
1363 SB 203580 MAPK inhibitor (p38 specific) €95.00
1364 SB 202190 MAPK inhibitor (p38 specific) €95.00
1365 PD169316 MAPK inhibitor (p38 specific) €95.00
1368 PD184352 MEK 1 inhibitor €80.00
1408 PD0325901 MEK1 and MEK2 inhibitor €50.00
1465 SB 203580 hydrochloride MAPK inhibitor (p38 specific) €70.00
1671 SCIO 469 MAPK inhibitor (p38 specific) €120.00
1694 FR 180204 ERK inhibitor; AP-1 inhibitor €95.00
1761 GSK 1120212 MEK1 and MEK2 inhibitor €70.00
1809 BIX 02189 MEK5 inhibitor; ERK5 inhibitor €110.00
1811 VX 745 Inhibitor of p38α MAP kinase €90.00
1837 PH 797804 Inhibitor of p38α MAPK €115.00
1846 XMD 8-92 BMK1 inhibitor; ERK5 inhibitor €70.00
1895 LY 2228820 Inhibitor of p38 MAPK €105.00
1999 AZD8330 MEK 1 inhibitor €105.00
1808 BIX02188-Me MEK5 inhibitor; ERK5 inhibitor €110.00
2366 NG 25 trihydrochloride Type II inhibitor of TAK1 (MAP3K7) and MAP4K2 (GCK) €75.00
2444 SB 706504 Selective p38 MAPK inhibitor that targets a subset of inflammatory macrophage genes. €125.00
2520 U 0126 Non-competitive inhibitor of MEK1/2 and protects brain in stroke models €90.00
2786 (±)-PH 797804 Inhibitor of p38α MAPK €115.00
3346 BIX02188 Potent MEK5 inhibitor €110.00
1621 XMD 8-92 trifluoroacetate BMK1 inhibitor; ERK5 inhibitor €70.00
3697 Binimetinib Potent, selective, non-ATP-competitive and orally available allosteric inhibitor of MEK1/2 €60.00
3874 RDEA119 Potent and highly selective small molecule allosteric MEK inhibitor Inquire

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Newsletter
Give Feedback
 
Send E-mail

Customer Support

About Axon Medchem

Download Product Catalog

Download the Axon Ligands™ catalogue 2021 Spring Edition

Follow Us

© 2016 Axon Medchem. All Rights Reserved.

Send us a message

×

Contact Us

* Required Fields

Please wait...