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FR 180204

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1694

CAS [865362-74-9]

MF C18H13N7
MW 327.34

  • Purity: 99%
  • Soluble in DMSO

FR 180204

Description

Selective, cell permeable and ATP-competitive ERK inhibitor; 30-fold selective on ERK over p38α MAPK; FR180204 was shown to inhibit ERK1 (Ki=0.31μM), ERK2 (Ki=0.14 μM) and TGFβ-induced AP-1 activation
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Size Unit Price Stock
5 mg €95.00 In Stock
10 mg €140.00 In Stock
50 mg €560.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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