Based on 1 reference(s) in Google Scholar 9 10 1

Axon 2680

CAS [1942114-09-1]

MW 383.40

  • Purity: 99%
  • Soluble in DMSO



EAI045 is an allosteric inhibitor that targets drug-resistant L858R/T790M-mutant EGFR tyrosine kinase (IC50 value of 3 nM), and spares the wild-type receptor (~1000-fold selectivity versus wild-type EGFR at 1 mM ATP).

KEYWORDS: EAI045 | supplier | Allosteric EGFR L858R/T790M inhibitor | EAI 045 | EAI-045 | CAS [1942114-09-1] | EGF | EGFR | Inhibitor | Receptors

Size Unit Price Stock
5 mg €105.00 In Stock
25 mg €375.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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