GSK 3787

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1628

CAS [188591-46-0]

MF C15H12ClF3N2O3S
MW 392.78

Purity: 99%
Soluble in DMSO

GSK 3787

Description

Selective and irreversible peroxisome proliferator-activated receptor (PPARδ) antagonist

PS Palkar et al. Cellular and Pharmacological Selectivity of the PPARβ/δ Antagonist GSK3787. Mol. Pharmacol. Fast Forward. 2010.06.01.

BG Shearer et al. Identification and characterization of 4-chloro-N-(2-{[5-trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide (GSK3787), a selective and irreversible PPARdelta antagonist. J. Med. Chem. 2010, 53(4), 1857-61.

PPARδ antagonist

Chemical name

4-chloro-N-(2-(5-(trifluoromethyl)pyridin-2-ylsulfonyl)ethyl)benzamide

Parent CAS No.

[188591-46-0]

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GSK 3787

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GSK 3787

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