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Xevinapant - AT-406 | DEBIO1143 | SM-406

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1985

CAS [1071992-99-8]

MF C32H43N5O4
MW 561.71

  • Purity: 100%
  • Optical purity: Optically pure
  • Soluble in DMSO

Xevinapant

Description

Potent and orally available antagonist of the inhibitor of apoptosis proteins (IAPs); binds to XIAP, cIAP1, and cIAP2 proteins with Ki of 66.4, 1.9, and 5.1 nM, respectively
Antagonist of Inhibitor of apoptosis proteins (IAPs)

Chemical name

(5S,8S,10aR)-N-benzhydryl-5-((S)-2-(methylamino)propanamido)-3-(3-methylbutanoyl)-6-oxodecahydropyrrolo[1,2-a][1,5]diazocine-8-carboxamide

Parent CAS No.

[1071992-99-8]

Order
Size Unit Price Stock
5 mg €145.00 In Stock
25 mg €505.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €220.00 In Stock
2 x 25 mg €760.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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