Kinases (OH-acceptors)
Enzymes are capable of transferring phosphate groups to an alcohol moiety of the acceptor substrate (EC 2.7.1.)
| Axon ID | Name | Description | From price | |
|---|---|---|---|---|
| 2175 | 3PO | Inhibitor of HIF-1-induced PFKFB3, an enzyme with a key role in glycolysis. | €65.00 | |
| 1831 | A 66 | PI3K inhibitor (p110-α specific) | €95.00 | |
| 2880 | ABC294640 | Selective and orally available SphK2 (or SK2) inhibitor | €125.00 | |
| 2289 | ABT 702 | The first, non-nucleoside adenosine kinase (ADK) inhibitor | €120.00 | |
| 2857 | Acalisib | PI3K inhibitor (p110 δ specific) | €120.00 | |
| 2925 | Alpelisib | PI3K inhibitor (p110-α specific) | €90.00 | |
| 1424 | AS 252424 | PI3K inhibitor (p110-γ specific) | €85.00 | |
| 1436 | AS 252424 bispotassium salt | PI3K inhibitor (p110-γ specific) | €95.00 | |
| 2748 | Autophinib | PIK3C3/Vps34 inhibitor | €120.00 | |
| 2926 | AZD 6482 | PI3K inhibitor (p110 β specific) | €120.00 | |
| 3062 | AZD1656 | Glucokinase (GK) activator | €165.00 | |
| 3690 | AZD8186 | PI3Kβ/δ isoform-selective inhibitor | Inquire | |
| 3055 | B591 | Potent, specific class I PI3K inhibitor | €125.00 | |
| 1282 | BAG 956 | PI3K and PDPK1 inhibitor | €95.00 | |
| 3357 | BAMB-4 | Membrane permeable ITPKA inhibitor (InsP3Kinase specific) | €120.00 | |
| 3598 | BAY-091 hydrochloride | First potent and highly selective PIP4K2A inhibitor | Recently added | €180.00 |
| 1281 | BEZ 235 | PI3K and mTOR tyrosine kinase inhibitor | €50.00 | |
| 2801 | BQR695 | PI4K inhibitor | €105.00 | |
| 2170 | CAL 101 | PI3K inhibitor (p110 δ specific) | €95.00 | |
| 2992 | CTx-0294885 | Broad-spectrum kinase inhibitor | €90.00 | |
| 2039 | CZC 24832 | PI3K inhibitor (p110-γ specific) | €95.00 | |
| 1719 | D 106669 | Potent and selective PI3K inhibitor | €85.00 | |
| 1377 | GDC 0941 bismesylate | PI3K inhibitor | €85.00 | |
| 1782 | GDC 0980 | Dual PI3K and mTOR inhibitor | €80.00 | |
| 2994 | GNE 317 | Brain-penetrant PI3K inhibitor (p110-α specific) | €85.00 | |
| 3434 | GNF362 | Potent, selective and orally bioavailable Itpkb inhibitor | €150.00 | |
| 1596 | GSK 2126458 | Dual PI3K and mTOR inhibitor | €50.00 | |
| 1912 | GSK 2636771 dihydrochloride | PI3K inhibitor (p110 β specific) | €105.00 | |
| 2168 | IC 87114 | Potent and highly selective inhibitor of the PI3K p110δ | €85.00 | |
| 2235 | K 145 hydrochloride | Selective, substrate competitive SphK2 inhibitor | €105.00 | |