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ML252

Axon 2615
  • Parent CAS:  1392494-64-2
Purity:  99%
  • Soluble in DMSO
  • MF:  C20H24N2O.HCl
  • MW:  344.88

Description

Potent, selective and brain penetrant KCNQ2 inhibitor (Kv7.2; IC50 value 69 nM, and >40-fold selective over KCNQ1). A useful in vivo tool molecule to study KCNQ2 pharmocology.

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