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XEN1101

 - Azetukalner
Axon 4428
CAS:  1009344-33-5
Purity:  99%
  • Soluble in DMSO and EtOH
  • MF:  C23H29FN2O
  • MW:  368.49

Description

XEN1101 is a second generation orally active Kv7 channel opener which was found to be ~4-fold selective for Kv7.2/7.3 over Kv7.3/7.5 and Kv7.4 channels, with EC 50 values of 27 nM versus 94 nM and 113 nM, respectively.

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