AG 014699 - PF 01367338 | Rucaparib

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1529

CAS [459868-92-9]

MF C19H18FN3O.H3O4P
MW 421.36

  • Purity: 98%
  • Soluble in water and DMSO

AG 014699

Description

A PARP 1 inhibitor with potential chemosensitizing, radiosensitizing and antineoplastic activities; selectively binds to PARP1 (Ki=1.4 nM) and inhibits PARP1-mediated DNA repair, thereby enhancing the accumulation of DNA strand breaks and promoting genomic instability and apoptosis. AG-014699 is the phosphate salt of AG 014447 (CAS 283173-50-2) and has improved aqueous solubility The camsylate salt form of Rucaparib is also available as Axon 3113.

KEYWORDS: AG 014699 | supplier | 283173-50-2 | 459868-92-9 | Axon 1529 | PARP1 inhibitor | Axon Ligands | Supplier | PF 01367338 | Axon1529 | AG014699 | PF01367338 | PARP1

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Size Unit Price Stock
2 mg €60.00 In Stock
5 mg €90.00 In Stock
25 mg €270.00 In Stock
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2 x 5 mg €130.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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