PDK1 inhibitor 2610

Based on 2 reference(s) in Google Scholar 8 10 2

Axon 2610

CAS [N.A.]

MF C25H15N5.HCl
MW 421.88

  • Purity: 99%
  • Soluble in water and DMSO

PDK1 inhibitor 2610

Description

Potent, ATP-competitive and selective dual PI3K and PDPK1 inhibitor (IC50 values 34 nM and 94 nM for PDK1 and p-T308-PKB inhibition, respectively. Also inhibits PI3K p110α, p110β, p110δ, and p110γ (IC50 values 64 nM, 432 nM , 98 nM, and 67 nM, respectively).

Axon 2610 is a close analogue of NVP-BAG956 (Axon 1282)

KEYWORDS: PDK1 inhibitor 2610 | supplier | PI3K/PDK1 inhibitor | CAS [853909-77-0] | Phosphatidylinositol | PI3K | PDPK | Inhibitor | PKB | Akt | p110 | Oncology | PIP3 | Novartis

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Size Unit Price Stock
5 mg €125.00 In Stock
25 mg €435.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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