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Axon 2486
CAS [1680193-80-9]
MF C22H20ClN5OMW 405.88
Selective reversible inhibitor of monoacylglycerol lipase (MAGL; IC50 value 46 nM) with 35-fold higher selectivity over human α/β-hydrolase-6 (ABHD6) and 150-fold higher selectivity over human FAAH. The Loratidine analog JZP 361 fully retained H1 antagonistic activity as well (pA2 value 6.81) but is devoid of cannabinoid receptor (CB) affinity.
KEYWORDS: JZP 361 | Supplier | MAGL inhibitor - H1 antagonist | JZP361 | CAS [1680193-80-9] | 2-arachidonoyl glycerol (2-AG) | MAGL | Inhibitor | antagonist | monoacylglycerol | lipase | histamine | allergy | Fatty acid amide hydrolase | FAAH | ABHD6
[4-(8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)-1-piperidinyl]-1H-1,2,4-triazol-1-yl-methanone
[1680193-80-9]
The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.
Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!
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