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L 002 - NSC 764414

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2319

CAS [321695-57-2]

MF C15H15NO5S
MW 321.35

  • Purity: 99%
  • Soluble in DMSO

L 002

Description

Inhibitor of p300 histone acyltransferase (a.k.a KAT3B; IC50 value 1.98 μM in vitro) that also inhibited acetylation of histones and p53, and suppresses STAT3 activation in cell-based assays. In vivo, L 002 potently suppressed tumor growth of TNBC cell line MDA-MB-468 xenografts.
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10 mg €80.00 In Stock
50 mg €280.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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