GSK J1

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 1934

CAS [1373422-53-7]

MF C22H23N5O2
MW 389.45

  • Purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO

GSK J1

Description

The first selective and potent histone demethylase JMJD3/UTX inhibitor; blocks demethylation of histone H3K27; showed no activity against a panel of JMJ family demethylases and 100 protein kinases.Available also a cell permeable ethyl ester derivative GSK J4 (Axon 1933), which is a prodrug suitable for cell-based studies and will be hydrolyzed to GSK-J1 in cells rapidly

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Size Unit Price Stock
5 mg €105.00 In Stock
25 mg €365.00 In Stock
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Size Unit Price Stock
2 x 5 mg €160.00 In Stock
2 x 25 mg €560.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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