AM 251

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1218

CAS [183232-66-8]

MF C22H21Cl2IN4O
MW 555.24

  • Purity: 99%
  • Soluble in DMSO and Ethanol

AM 251


Cannabinoids CB1 antagonist, structurally very close to SR 141716A (rimonabant). AM251: Ki 7.5 nM for CB1 receptor vs SR 141716A ( Ki value of 11.5 nM). However AM251 is about two-fold more selective for the CB1 receptor when compared to SR 141716A
Size Unit Price Stock
10 mg €95.00 In Stock
50 mg €285.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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