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GAT211
- Soluble in DMSO and EtOH
- MF: C22H18N2O2
- MW: 342.39
Description
GAT211 is a potent CB1 receptor ago-PAM with allosteric agonist activity residing exclusively in the R-(+)-enantiomer, GAT228 (Axon 4358), and S-(-)-enantiomer, GAT229 (Axon 4359), acting as a “pure” and potent CB1R PAM. GAT211 engages CB1R allosteric site(s), enhances the binding of the orthosteric full agonist [3H]CP55,490, and reduces the binding of the orthosteric antagonist/inverse agonist [3H]SR141716A.
KEYWORDS: GAT211 | Supplier | CB1 ago-PAM | GAT-211 | GAT 211 | CAS [102704-40-5] | Cannabinoids | CB1 | Agonist | PAM | Receptors
More Information
| Parent CAS No. | 102704-40-5 |
|---|---|
| Chemical Name | 3-(2-Nitro-1-phenylethyl)-2-phenylindole |
| Short Description | CB1 ago-PAM |
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