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Receptors
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Opioid
OPR-μ
Naloxonazine dihydrochloride

Naloxonazine dihydrochloride - NSC 612113

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1205

CAS [880759-65-9]

MF C38H42N4O6.2HCl
MW 723.69

Purity: 97%
Soluble in water

Naloxonazine dihydrochloride

Description

Naloxonazine dihydrochloride is a potent opioid antagonist, selective for μ1 receptors.

KEYWORDS: Naloxonazine dihydrochloride | Supplier | 82824-01-9 | 880759-65-9 | Opioid antagonist | Axon Ligands | NSC 612113 | Naloxonazine | NSC612113 | OPR-μ

D Paul et al. Differential blockade by naloxonazine of two mu opiate actions: analgesia and inhibition of gastrointestinal transit. Eur J Pharmacol. 1988 May 10;149(3):403-4.

CC Chien et al. Naloxonazine, a specific mu-opioid receptor antagonist, attenuates the increment of locomotor activity induced by acute methamphetamine in mice. Toxicol Lett. 2012 Jul 7;212(1):61-5.

EF Hahn et al. Naloxonazine, a potent, long-lasting inhibitor of opiate binding sites. Life Sci. 1982 Sep 20-27;31(12-13):1385-8.

G De Muylder et al. Naloxonazine, an Amastigote-Specific Compound, Affects Leishmania Parasites through Modulation of Host-Encoded Functions. PLoS Negl Trop Dis. 2016 Dec 30;10(12):e0005234.

Cell Signaling & Oncology CNS Pain & Inflammation Endocrinology OPR-μ A4

Opioid antagonist

Chemical name

4,5-epoxy-3,14-dihydroxy-17-(2-propen-1-yl)-, 2-[(5a)-4,5-epoxy-3,14-dihydroxy-17-(2-propen-1-yl)morphinan-6-ylidene]hydrazone-morphinan-6-one dihydrochloride

Parent CAS No.

[82824-01-9]

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Size	Unit Price	Stock
10 mg	€120.00	In Stock
50 mg	€450.00	In Stock

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