JavaScript seems to be disabled in your browser.
You must have JavaScript enabled in your browser to utilize the functionality of this website.

Axon Medchem

All

Home
Products
- Shop By Category
- Featured Products
- Shop By Alphabet
  - A
  - B
  - C
  - D
  - E
  - F
  - G
  - H
  - I
  - J
  - K
  - L
  - M
  - N
  - O
  - P
  - Q
  - R
  - S
  - T
  - U
  - V
  - W
  - X
  - Y
  - Z
  - #
Support
- - Customer Support
  - Customer Services
Contact
- About Axon Medchem
- Contact Us

Home
Products
Receptors
GPCR
Opioid
OPR-μ
Naloxonazine dihydrochloride

Naloxonazine dihydrochloride - NSC 612113

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1205

CAS [880759-65-9]

MF C38H42N4O6.2HCl
MW 723.69

Purity: 97%
Soluble in water

Naloxonazine dihydrochloride

Description

Naloxonazine dihydrochloride is a potent opioid antagonist, selective for μ1 receptors.

KEYWORDS: Naloxonazine dihydrochloride | Supplier | 82824-01-9 | 880759-65-9 | Opioid antagonist | Axon Ligands | NSC 612113 | Naloxonazine | NSC612113 | OPR-μ

D Paul et al. Differential blockade by naloxonazine of two mu opiate actions: analgesia and inhibition of gastrointestinal transit. Eur J Pharmacol. 1988 May 10;149(3):403-4.

CC Chien et al. Naloxonazine, a specific mu-opioid receptor antagonist, attenuates the increment of locomotor activity induced by acute methamphetamine in mice. Toxicol Lett. 2012 Jul 7;212(1):61-5.

EF Hahn et al. Naloxonazine, a potent, long-lasting inhibitor of opiate binding sites. Life Sci. 1982 Sep 20-27;31(12-13):1385-8.

G De Muylder et al. Naloxonazine, an Amastigote-Specific Compound, Affects Leishmania Parasites through Modulation of Host-Encoded Functions. PLoS Negl Trop Dis. 2016 Dec 30;10(12):e0005234.

Cell Signaling & Oncology CNS Pain & Inflammation Endocrinology OPR-μ A4

Opioid antagonist

Chemical name

4,5-epoxy-3,14-dihydroxy-17-(2-propen-1-yl)-, 2-[(5a)-4,5-epoxy-3,14-dihydroxy-17-(2-propen-1-yl)morphinan-6-ylidene]hydrazone-morphinan-6-one dihydrochloride

Parent CAS No.

[82824-01-9]

Order

Size	Unit Price	Stock
10 mg	€130.00	In Stock
50 mg	€490.00	In Stock

Need more? Bulk Inquiry

Related Products

Axon ID	Name	Description	From price
1140	Fedotozine tartrate	Kappa(1a) opioid agonist		€135.00
1163	nor-Binaltorphimine dihydrochloride	Kappa-opioid antagonist		Inquire
1202	U-50488 hydrochloride	Kappa-opioid agonist		€80.00
1213	β-Funaltrexamine hydrochloride	Mu-opioid antagonist		€90.00
1230	Naloxone Benzoylhydrazone	Kappa-opioid agonist		€90.00
1412	SNC 80	δ-opioid agonist		€120.00
1413	SB 612111 hydrochloride	NOP antagonist		€80.00
1573	Nalmefene hydrochloride	Opioid antagonist		€90.00
1577	Nalbuphine hydrochloride	Analgesic. Κ-opioid agonist and μ-opioid antagonist/partial agonist		€140.00
1751	ADL 5859	Selective δ-opioid receptor agonist		€115.00
1784	BAN ORL 24 dihydrochloride	NOP receptor antagonist		Inquire
1805	JTC 801	NOP receptor antagonist		€90.00
2415	Naloxone hydrochloride	Neutral opioid antagonist		€50.00
2416	Naltrexone hydrochloride	Competitive opioid antagonist with preference for µ- and κ-receptors		€60.00
1226	GNTI dihydrochloride	Kappa-opioid antagonist		€160.00
3640	Loperamide hydrochloride	Potent Mu-opioid agonist		€50.00

Please wait...