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Muzepan1
- Soluble in DMSO
- MF: C21H22BrCl2N3O
- MW: 483.23
Description
Muzepan1 is a brain-penetrant Mu (μ) opioid receptor (MOR) agonist (pEC50 value of 7.06) with having state-selective affinity for promoting GTP release versus GTP binding.
More Information
| Parent CAS No. | N.A. |
|---|---|
| Chemical Name | 1-(1-(1-(4-Bromophenyl)ethyl)-4-azepanyl)-5,6-dichloro-1,3-dihydro-2H-1,3-benzimidazol-2-one |
| Short Description | Mu-opioid agonist |
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