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Muzepan1

Axon 4456
CAS:  N.A.
Purity:  98%
  • Soluble in DMSO
  • MF:  C21H22BrCl2N3O
  • MW:  483.23

Description

Muzepan1 is a brain-penetrant Mu (μ) opioid receptor (MOR) agonist (pEC50 value of 7.06) with having state-selective affinity for promoting GTP release versus GTP binding.

More Information

Parent CAS No. N.A.
Chemical Name 1-(1-(1-(4-Bromophenyl)ethyl)-4-azepanyl)-5,6-dichloro-1,3-dihydro-2H-1,3-benzimidazol-2-one
Short Description Mu-opioid agonist

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