Based on 10 reference(s) in Google Scholar 8 10 10

Axon 2790

CAS [56632-39-4]

MF C21H17NO3
MW 331.36

  • Purity: 99%
  • Soluble in 0.1N NaOH(aq) and DMSO



BHPI is a potent noncompetitive ERα inhibitor that selectively blocks proliferation of drug-resistant ERα-positive breast and ovarian cancer cells (IC50 values of 27 and 15 nM in MDA-468 and T47D cell lines, respectively). Moreover, BHPI induced rapid and substantial tumor regression in a mouse xenograft model of breast cancer.

KEYWORDS: BHPI | supplier | ER-α antagonist | CAS [56632-39-4] | Estrogen | Estrogen (ER) | Antagonist | Receptors | Breast cancer

Size Unit Price Stock
10 mg €125.00 In Stock
50 mg €475.00 In Stock
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Size Unit Price Stock
2 x 10 mg €200.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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