LW6

Based on 62 publications in PubMed 9 10 62

Axon 2480

CAS [934593-90-5]

MF C26H29NO5
MW 435.51

  • Purity: 99%
  • Soluble in DMSO

LW6

Description

Novel HIF-1 inhibitor (IC50 value 2.44 μM) that promotes proteasomal degradation of HIF-1α via upregulation of von-Hippel-Lindau (VHL), without affecting the activity of prolyl hydroxylase (PHD). Evidence was found that identified MDH2 as a target protein of LW-6. Moreover, LW6 suppresses angiogenesis by inhibition of HIF-1α stability via direct binding with calcineurin b homologous protein 1 (CHP1) in a Ca2+ dependent manner.

KEYWORDS: LW 6 | supplier | HIF-1 inhibitor | LW6 | CAS [934593-90-5] | DNA-RNA | HIF-1 | CHP1 | Inhibitor | Transcription Factor | hypoxia inducible factor | angiogenesis | tumor | cancer | von-Hippel-Lindau | VHL | prolyl hydroxylase | PHD | calcineurin b homologous protein 1 | endoplasmic reticulum | malate dehydrogenase 2 | MDH2

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Size Unit Price Stock
10 mg €85.00 In Stock
50 mg €350.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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