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VU 0029767

Based on 12 reference(s) in Google Scholar 9 10 12

Axon 1988

CAS [326001-01-8]

MF C21H21N3O3
MW 363.41

  • Purity: 98%
  • Soluble in DMSO

VU 0029767

Description

Positive allosteric modulator of M1. VU 0029767 potentiates the agonistic effect of ACh for M1 (Ki value shifted by VU0029767 (3, 10 and 30 M) and shifted the ACh competition curve by 1.7 0.8-, 4.9 2.0-, and 8.8 1.9-fold, respectively, compared to control (DMSO; Ki value 8.7 µM). VU0029767 potentiates ACh-mediated intracellular calcium mobilization, but not phospholipase D activation.
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Size Unit Price Stock
10 mg €110.00 In Stock
50 mg €390.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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