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Zamifenacin fumarate
- UK 76654
- Parent CAS: 127308-82-1
- Optical Purity: >98% e.e.
- Soluble in DMSO and EtOH
- MF: C31H33NO7
- MW: 531.6
Description
Zamifenacin fumarate is a selective M3 muscarinic acetylcholine receptor antagonist.
M3 receptors regulate smooth muscle contraction, glandular secretion and cholinergic responses in bladder, airway and gastrointestinal tissues. Zamifenacin is useful for evaluating M3 receptor blockade and muscarinic subtype selectivity.
Key Features
- Selective M3 muscarinic receptor antagonist
- Blocks CHRM3-mediated cholinergic signaling
- Relevant to smooth muscle and secretory responses
- Useful for muscarinic receptor subtype profiling
Applications
- M3 receptor binding and functional assays
- Bladder and gastrointestinal smooth muscle studies
- Cholinergic signaling research
- Muscarinic antagonist selectivity profiling
More Information
| Parent CAS No. | 127308-82-1 |
|---|---|
| Chemical Name | (R)-3-Benzhydryloxy-1-(2-benzo[1,3]dioxol-5-yl-ethyl)-piperidine fumarate |
| SMILES | C1(CCN2CCC[C@@H](OC(C3C=CC=CC=3)C3C=CC=CC=3)C2)C=C2OCOC2=CC=1.C(/C(=O)O)=CC(=O)O |&1:7,r| |
| MFCD | N.A. |
| InChi | InChI=1S/C27H29NO3.C4H4O4/c1-3-8-22(9-4-1)27(23-10-5-2-6-11-23)31-24-12-7-16-28(19-24)17-15-21-13-14-25-26(18-21)30-20-29-25;5-3(6)1-2-4(7)8/h1-6,8-11,13-14,18,24,27H,7,12,15-17,19-20H2;1-2H,(H,5,6)(H,7,8)/b;2-1+/t24-;/m1./s1 |
| InChiKey | PMHKTAIGYOVZEZ-ZHWJIHCSSA-N |
| CID | 20056967 |
| Short Description | M3 antagonist |
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