Elacestrant dihydrochloride - RAD1901

Based on 43 reference(s) in Google Scholar 8 10 43

Axon 4095

CAS [1349723-93-8]

MF C30H38N2O2.2HCl
MW 531.56

  • Purity: 99%
  • Optical purity: 100% e.e.
  • Soluble in water and DMSO

Elacestrant dihydrochloride

Description

Elacestrant dihydrochloride is an orally bioavailable selective estrogen receptor degrader (SERD) with IC50 values of 48 nM and 870 nM for ERα and ERβ, respectively. Elacestrant is a potent antagonist of breast cancer cells, inhibiting both basal and E2-stimulated MCF-7 cell proliferation.

Keywords: Elacestrant dihydrochloride | Supplier | SERD | RAD1901 | RAD 1901 | RAD-1901 | Orserdu | CAS [1349723-93-8] | [722533-56-4] | Estrogen | Estrogen (ER) | Degrader | Receptors | Breast cancer | Postmenopausal | SERM

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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

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