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Vorasidenib - AG881

Based on 18 reference(s) in Google Scholar 8 10 18

Axon 4024

CAS [1644545-52-7]

MF C14H13ClF6N6
MW 414.74

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in DMSO and EtOH

Vorasidenib

Description

Vorasidenib is a first-in-class, potent, orally active, brain-penetrant dual mIDH1/2 inhibitor with IC50 values of 6 nM and 12 nM for IDH1-R132H and IDH2-R140Q, respectively.

Keywords: Vorasidenib | Supplier | IDH1/2 inhibitor | AG881 | AG 881 | AG-881 | CAS [1644545-52-7] | Isocitrate | IDH | Inhibitor | Enzymes | Glioma

First-in-class, potent, orally active, brain-penetrant dual mIDH1/2

Chemical name

6-(6-Chloropyridin-2-yl)-N2,N4-bis((R)-1,1,1-trifluoropropan-2-yl)-1,3,5-triazine-2,4-diamine

Parent CAS No.

[1644545-52-7]

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Size Unit Price Stock
10 mg €140.00 In Stock
50 mg €520.00 In Stock
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3863 BAY-1436032 Highly selective, potent and orally available inhibitor of mutant Isocitrate Dehydrogenase 1 (mIDH1) Inquire

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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