MC4171

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 4011

CAS [3034769-78-0]

MF C21H15N3O3
MW 357.37

  • Purity: 98%
  • Soluble in 0.1N NaOH(aq), DMSO and EtOH
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MC4171

Description

MC4171 is a first-in-class potent and selective inhibitor of the lysine acetyltransferase KAT8 with an IC50 value of 8.1 μM. Moreover, MC4171 exhibited mid-micromolar antiproliferative activity in different cancer cell lines, including NSCLC and AML, without impacting the viability of nontransformed cells.

KEYWORDS: MC4171 | Supplier | KAT8 inhibitor | MC 4171 | MC-4171 | CAS [3034769-78-0] | Histone | HAT | Inhibitor | Enzymes | MOF | MYST1 | Cancer

First-in-class potent and selective KAT8 inhibitor

Chemical name

(Z)-4-(4-((1H-Pyrrol-2-yl)methylene)-5-oxo-3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)benzoic acid

Parent CAS No.

[3034769-78-0]

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Size Unit Price Stock
10 mg €130.00 In Stock
50 mg €520.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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