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KDM5 inhibitor compound 48

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 2809

CAS [1628210-26-3]

MF C17H20N6O
MW 324.38

  • Purity: 99%
  • Soluble in DMSO

KDM5 inhibitor compound 48

Description

Potent, selective and orally bioavailable KDM5 inhibitor (IC50 value of 15.1 nM for KDM5A) with improved cell potency (EC50 value of 0.34 μM, H3K4Me3 level in PC9 cells). Chemical probe suitable for studying KDM5 biological functions in vivo.

KEYWORDS: KDM5 inhibitor compound 48 | supplier | KDM5 inhibitor | CAS [1628210-26-3] | Histone demethylase | Inhibitor | Enzymes | Orally bioavailable | PC9

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5 mg €145.00 In Stock
25 mg €505.00 In Stock
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2 x 5 mg €230.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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