SB 332235

Based on 62 reference(s) in Google Scholar 9 10 62

Axon 2593

CAS [276702-15-9]

MF C13H10Cl3N3O4S
MW 410.66

  • Purity: 98%
  • Soluble in 0.1N NaOH(aq) and DMSO

SB 332235

Description

Selective nonpeptide CXCR2 antagonist (IC50 values 9.3 nM and 9.6 µM for CXCR2 and CXCR1, respectively) exhibiting significant anti-inflammatory effects in acute and chronic models of arthritis in the rabbit. SB-332235 significantly reduced levels of proinflammatory mediators in the synovial fluid, including TNF-α, IL-8, PGE2, LTB4, and LTC4. SB-332235 was also found to abolish the GRO/CINC-1 mediated inhibition of C2-ceramide-induced cytochrome-c release from mitochondria.

KEYWORDS: SB 332235 | supplier | CXCR2 antagonist | SB332235 | SB-332235 | CAS [276702-15-9] | Chemokine | GPCR | anti-inflammatory | arthritis |  TNF-α | IL-8 | interleukin-8 | PGE2 | prostaglandin | LTB4 | LTC4 | Alzheimer's | apoptosis

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Size Unit Price Stock
5 mg €105.00 In Stock
25 mg €365.00 In Stock
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Size Unit Price Stock
2 x 5 mg €160.00 In Stock
2 x 25 mg €580.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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