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PPQ 102

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2295

CAS [931706-15-9]

MF C26H22N4O3
MW 438.48

  • Purity: 99%
  • Soluble in DMSO

PPQ 102

Description

Potent CFTR inhibitor (IC50 value ca 90 nM in CFTR chloride conductance essay). PPQ 102 acts by a mechanism involving stabilization of the channel closed-state. Prevented cyst expansion and reduced the size of preformed cysts in an embryonic kidney organ culture model of Polycystic kidney disease (PKD).
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Size Unit Price Stock
5 mg €100.00 In Stock
25 mg €360.00 In Stock
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2 x 5 mg €160.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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