VU 0255035 - ML012

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1787

CAS [1135243-19-4]

MF C18H20N6O3S2
MW 432.52

VU 0255035

Description

Highly selective antagonist of M1 muscarinic acetylcholine receptor (mAChR) (Ki=14.87 nM).

CNS CHRM1 A18

Selective M1 mAChR Antagonist

N-(3-oxo-3-(4-(pyridin-4-yl)piperazin-1-yl)propyl)benzo[c][1,2,5]thiadiazole-4-sulfonamide

[1135243-19-4]

Order

Size	Unit Price	Stock
10 mg	€120.00	In Stock
50 mg	€480.00	In Stock

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Axon ID	Name	Description
1109	Etiracetam	Racemate of Axon 1110 and Axon 1111	€75.00
1110	Levetiracetam	Binds synaptic vesicle protein 2A (SV2A)	€85.00
1111	UCB-L 060	Least active enantiomer of Axon 1109	€120.00
1273	Zamifenacin fumarate	Muscarinic M3 antagonist	€130.00
1483	VU 0152100	PAM of M4 mAChR	€85.00
1679	MDL 201012	Muscarinic M3 antagonist	€110.00
1703	VU 0357017 hydrochloride	PAM of M1 mAChR	€115.00
1786	VU 0238429	Selective PAM of M5 mAChR (CHRM5)	€105.00
1943	VU 0365114	Selective PAM of M5 mAChR (CHRM5)	€115.00
2049	Tolterodine L-tartrate	Muscarinic receptor (mAChR) antagonist	€60.00
1988	VU 0029767	PAM of mAChR M1 that potentiates the agonistic effect of Ach	€110.00
2463	TBPB	Allosteric activator of the M1 acetylcholine receptor devoid of M2-M5 activity.	€105.00
2587	ML352	Potent and selective inhibitor of the presynaptic choline transporter CHT	€105.00
2670	VU6001221	Choline transporter inhibitor	€125.00
3271	VU0486846	Potent and highly selective PAM of M1 mAChR	€165.00
3286	Penehyclidine hydrochloride	Anticholinergic drug	€130.00
3505	Oxybutynin hydrochloride	Competitive M1/M2/M3 mAChR antagonist	€50.00
3513	Bethanechol chloride	Muscarinic receptor (mAChR) agonist	€50.00
3648	Trospium chloride	Specific, orally active and competitive muscarinic receptor (mAChR) antagonist	€60.00