BI-D1870

Based on 177 publications in PubMed 9 10 177

Axon 1528

CAS [501437-28-1]

MF C19H23F2N5O2
MW 391.42

  • Purity: 99%
  • Soluble in DMSO and Ethanol

BI-D1870

Description

Potent and specific inhibitor of the p90 ribosomal S6 kinase (RSK) isoforms in vitro and in vivo, which inhibits RSK1, RSK2, RSK3 and RSK4 in vitro (IC50 values 31 nM, 24 nM, 18 nM, and 15 nM, respectively).
* BI-D1870 binds at NTKD binding site as a reversible RSK inhibitor, while FMK (Axon 1848) binds at CTKD site as an irreversible RSK inhibitor.  

KEYWORDS: BI-D1870 | supplier | RSK inhibitor | BID1870 | BID-1870 | CAS [501437-28-1] | p90-RSK | p90 ribosomal S6 kinase | RSK1 | RSK2 | RSK3 | RSK4 | NTKD binding site | reversible

Order
Size Unit Price Stock
2 mg €80.00 In Stock
5 mg €105.00 In Stock
25 mg €365.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €160.00 In Stock
2 x 25 mg €560.00 In Stock
Need more? Bulk Inquiry

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Please wait...