GSK J4

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1933

CAS [1373423-53-0]

MF C24H27N5O2
MW 417.50

  • Purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO

GSK J4

Description

Histone demethylase JMJD3/UTX inhibitor; blocks demethylation of histone H3K27; As a cell permeable ethyl ester derivative of GSK J1 (Axon 1934), it is a suitable prodrug form for cell-based studies. It is rapidly hydrolyzed in cells, generateing pharmacologically relevant intracellular concentrations of GSK-J1

Order
Size Unit Price Stock
5 mg €105.00 In Stock
25 mg €365.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €160.00 In Stock
2 x 25 mg €560.00 In Stock
Need more? Bulk Inquiry

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Please wait...