GSK-LSD1

Based on 14 reference(s) in Google Scholar 8 10 14

Axon 2375

CAS [N.A.]

MF C14H20N2.2HCl
MW 289.24

  • Purity: 99%
  • Optical purity: mixture of trans-diastereomers
  • Soluble in water and DMSO

GSK-LSD1

Description

Irreversible inhibitor of the KDM1 family histone demethylase LSD1 (IC50 value 16 nM). GSK-LSD1 is >1000 fold selective over closely related FAD utilizing enzymes (i.e. LSD2, MAO-A, MAO-B), induces gene expression changes in cancer cell lines (average EC50 <5 nM), and inhibits cancer cell line growth (average EC50 <5 nM).
Order
Size Unit Price Stock
10 mg €110.00 In Stock
50 mg €420.00 In Stock
Special Offers
Size Unit Price Stock
2 x 10 mg €180.00 In Stock
Need more? Bulk Inquiry

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Please wait...