Loperamide hydrochloride

Based on 2221 reference(s) in Google Scholar 8 10 2221

Axon 3640

CAS [34552-83-5]

MF C29H33ClN2O2.HCl
MW 513.50

  • Purity: 100%
  • Soluble in DMSO and EtOH

Loperamide hydrochloride


Loperamide is a peripherally restricted potent μ-opioid receptor (MOR) agonist with a Ki value of 3.3 nM. Loperamide can also inhibit voltage-gated L-type calcium channels and trigger autophagy-dependent cell death as well. Antidiarrheal medicine.

KEYWORDS: Loperamide hydrochloride | Supplier | u-opioid agonist | R18553 | Imodium | CAS [34552-83-5] | [53179-11-6] | Opioids | OPR-μ | Agonist | Receptors

Potent Mu-opioid agonist

Chemical name

4-(4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl)-N,N-dimethyl-2,2-diphenylbutanamide hydrochloride

Parent CAS No.


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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

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