SUVN-502 is a potent, selective and orally active serotonin 6 (5-HT6) receptor antagonist (Ki value of 2.04 nM) with selectivity over 100 target sites which include receptors, enzymes, peptides, growth factors, ion channels, steroids, immunological factors, second messengers, and prostaglandins. Moreover, it has high selectivity over 5-HT2A receptor. SUVN-502 is brain penetrant and a clinical candidate for potential treatment of cognitive disorders.

KEYWORDS: SUVN-502 | supplier | 5-HT6 antagonist | SUVN502 | SUVN 502 | CAS [1791396-46-7] | [701205-60-9] | Serotonin | 5-HT6 | Antagonist | Receptors | Alzheimer