OTX 015

Based on 345 reference(s) in Google Scholar 10 10 345

Axon 2530

CAS [202590-98-5]

MF C25H22ClN5O2S
MW 491.99

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in DMSO and ethanol

OTX 015

Description

Potent inhibitor of BRD2, BRD3, and BRD4 (Ki values ranging from 3.2 to 24.7 nM, considering BDs 1 and 2), with clear anti-proliferative activity on a large number of diffuse large B-cell lymphoma (DLBCL) cell lines. OTX 015 inhibits the growth of hematologic malignances through directly regulating MYC expression and activity.

KEYWORDS: OTX 015 | supplier | BET-BRD inhibitor | OTX015 | CAS [202590-98-5] | Histone | BET (BRD) | Inhibitor | BRD2 | BRD3 | BRD4 | tumor | apoptosis | G1 | cell cycle | diffuse large B-cell lymphoma | DLBCL | MYC

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Size Unit Price Stock
5 mg €125.00 In Stock
25 mg €435.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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