Your cart

There are no items in your shopping cart

VU 0365114

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1943

CAS [1208222-39-2]

MF C22H14F3NO3
MW 397.35

  • Purity: 99%
  • Soluble in DMSO and Ethanol

VU 0365114

Description

Selective positive allosteric modulator (PAM) of M5 muscarinic acetylcholine receptor (mAChR), with EC50 = 2.7 µM for M5 and >30 µM for M1–M4 subtypes
Order
Size Unit Price Stock
10 mg €115.00 In Stock
50 mg €345.00 In Stock
Need more? Bulk Inquiry

Related Products

Axon ID Name Description From price
1109 Etiracetam Racemate of Axon 1110 and Axon 1111 €75.00
1110 Levetiracetam Binds synaptic vesicle protein 2A (SV2A) €85.00
1111 UCB-L 060 Least active enantiomer of Axon 1109 €120.00
1273 Zamifenacin fumarate Muscarinic M3 antagonist €130.00
1483 VU 0152100 PAM of M4 mAChR €85.00
1679 MDL 201012 Muscarinic M3 antagonist €110.00
1703 VU 0357017 hydrochloride PAM of M1 mAChR €115.00
1786 VU 0238429 Selective PAM of M5 mAChR (CHRM5) €105.00
1787 VU 0255035 Selective M1 mAChR Antagonist €120.00
2049 Tolterodine L-tartrate Muscarinic receptor (mAChR) antagonist €60.00
1988 VU 0029767 PAM of mAChR M1 that potentiates the agonistic effect of Ach €110.00
2463 TBPB Allosteric activator of the M1 acetylcholine receptor devoid of M2-M5 activity. €105.00
2587 ML352 Potent and selective inhibitor of the presynaptic choline transporter CHT €105.00
2670 VU6001221 Choline transporter inhibitor €125.00
2739 VU 6008667 Selective NAM of M5 mAChR (CHRM5) €105.00
3286 Penehyclidine hydrochloride Anticholinergic drug €130.00
3513 Bethanechol chloride Muscarinic receptor (mAChR) agonist €50.00
3648 Trospium chloride Specific, orally active and competitive muscarinic receptor (mAChR) antagonist €60.00

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Newsletter
Give Feedback
 
Send E-mail

Customer Support

About Axon Medchem

Download Product Catalog

Download the Axon Ligands™ catalogue 2021 Spring Edition

Follow Us

© 2016 Axon Medchem. All Rights Reserved.

Send us a message

×

Contact Us

* Required Fields

Please wait...