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5-HT6 antagonist 29
Axon 1575
- Parent CAS: 478082-77-8
Purity:
99%
- Soluble in DMSO
- MF: C19H20ClN3O2S.HCl
- MW: 426.36
Description
Selective brain penetrant 5-HT6 receptor antagonist (pKi value 8.6). Close regio-isomer of SB 699929 with brain–blood ratio of 2.6:1 and ED50 value of 5 mg/kg (po), and thus twice as potent as SB 271046 (Axon 1099).
More Information
| Parent CAS No. | 478082-77-8 |
|---|---|
| Chemical Name | 3-(4-chlorophenylsulfonyl)-1-methyl-7-(piperazin-1-yl)-1H-indole hydrochloride |
| SMILES | C1C(N2CCNCC2)=C2N(C)C=C(S(C3C=CC(Cl)=CC=3)(=O)=O)C2=CC=1.Cl |
| MFCD | N.A. |
| InChi | InChI=1S/C19H20ClN3O2S.ClH/c1-22-13-18(26(24,25)15-7-5-14(20)6-8-15)16-3-2-4-17(19(16)22)23-11-9-21-10-12-23;/h2-8,13,21H,9-12H2,1H3;1H |
| InChiKey | MERMVFOBIFLWLA-UHFFFAOYSA-N |
| CID | 91826472 |
| Short Description | 5-HT6 antagonist |
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