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5-HT6 antagonist 29

Based on 18 reference(s) in Google Scholar 9 10 18

Axon 1575

CAS [497963-70-9]

MF C19H20ClN3O2S.HCl
MW 426.36

  • Purity: 99%
  • Soluble in DMSO

5-HT6 antagonist 29

Description

Selective brain penetrant 5-HT6 receptor antagonist (pKi value 8.6). Close regio-isomer of SB 699929 with brain–blood ratio of 2.6:1 and ED50 value of 5 mg/kg (po), and thus twice as potent as SB 271046 (Axon 1099).

Selective brain penetrant 5-HT6 receptor antagonist

Chemical name

3-(3-chlorophenylsulfonyl)-1-methyl-7-(piperazin-1-yl)-1H-indole hydrochloride

Parent CAS No.

[478082-77-8]

Order
Size Unit Price Stock
5 mg €90.00 In Stock
25 mg €300.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €140.00 In Stock
2 x 25 mg €460.00 In Stock
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Related Products

Axon ID Name Description From price
1099 SB 271046 hydrochloride 5-HT6 antagonist €95.00
1330 RO 04-6790 hydrochloride 5-HT6 antagonist €95.00
1382 SB 742457 hydrochloride 5-HT6 antagonist €80.00
1710 WAY 208466 dihydrochloride Potent and selective 5-HT6 receptor agonist €120.00
1849 MS 245 oxalate 5-HT6 antagonist €105.00
1927 SGS 518 Selective 5-HT6 antagonist €90.00
2144 Lu AE58054 hydrochloride Selective 5-HT6 antagonist with good oral bioavailability €90.00
2715 SUVN-502 Selective, orally active, brain-penetrant 5-HT6 receptor antagonist €105.00

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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