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GMC 1-116

Based on 15 reference(s) in Google Scholar 8 10 15

Axon 1151

CAS [63687-94-5]

MF C18H20N4O
MW 308.38

  • Purity: 99%
  • Soluble in 0.1N HCl(aq) and DMSO

GMC 1-116

Description

Analogue and metabolite of clozapine (Axon 1146); devoid of DA and α1 affinities, with weak 5-HT2 affinities but high M1 affinity (IC50=27 nM).

Another analogue and metabolite of cloazapine, with 2-Hydroxy moiety, GMC1-165 (Axon 1152), is also available.

KEYWORDS: GMC 1-116 | supplier | Clozapine analogue | GMC1-116 | CAS [63687-94-5] | Serotonin; Dopamine | D (Non Selective) | 5-HT (Non Selective) | Agonist | Receptors

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Size Unit Price Stock
5 mg €125.00 In Stock
25 mg €450.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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