Bulk Inquiry
PSB-0777
- Optical Purity: Optically pure
- Soluble in 0.1N NaOH(aq) and DMSO
- MF: C18H21N5O7S2
- MW: 483.52
Description
PSB-0777 is an adenosine A2A receptor agonist with a Ki value of 44.4 nM (rat brain striatum A2A receptor). PSB-0777 significantly improved impaired acetylcholine-induced contractions induced by 2,4,6-trinitrobenzenesulfonic acid and showed synergism with an A2B-selective antagonist. Its salt form, PSB-0777 ammonium salt (Axon 4377), is also available.
More Information
| Parent CAS No. | 1341190-47-3 |
|---|---|
| Chemical Name | 4-(2-(9-((2R,3R,4S,5R)-3,4-Dihydroxy-5-(hydroxymethyl)tetrahydro-2-furyl)-2-adenineylthio)ethyl)benzenesulfonic acid |
| SMILES | [C@H]1(N2C=NC3=C2N=C(SCCC2=CC=C(S(=O)(O)=O)C=C2)N=C3N)[C@H](O)[C@H](O)[C@@H](CO)O1 |&1:0,24,26,28,r| |
| MFCD | N.A. |
| InChi | InChI=1S/C18H21N5O7S2/c19-15-12-16(23(8-20-12)17-14(26)13(25)11(7-24)30-17)22-18(21-15)31-6-5-9-1-3-10(4-2-9)32(27,28)29/h1-4,8,11,13-14,17,24-26H,5-7H2,(H2,19,21,22)(H,27,28,29)/t11-,13-,14-,17-/m1/s1 |
| InChiKey | MSSJGFVZLYCDOA-LSCFUAHRSA-N |
| CID | 56838950 |
| Short Description | A2A agonist |
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