Bulk Inquiry
SB 242084
- Soluble in 0.1N HCl(aq), DMSO and EtOH
- MF: C21H19ClN4O2
- MW: 394.85
Description
Selective and brain penetrant 5-HT2C receptor antagonist. Its hydrochloride salt, SB 242084 hydrochloride, is available as Axon 1745.
More Information
| Parent CAS No. | 181632-25-7 |
|---|---|
| Chemical Name | 6-Chloro-5-methyl-N-(6-(2-methylpyridin-3-yloxy)pyridin-3-yl)indoline-1-carboxamide |
| MFCD | N.A. |
| Short Description | 5-HT2C antagonist |
References
- SM Bromidge et al. 6-Chloro-5-methyl-1-[[(2-methyl-3-pyridyl)oxy]-5-pyridyl]carbamoyl]-indoline (SB-242084): the first selective and brain penetrant 5-HT2C receptor antagonist. J. Med. Chem. 1997, 40(22), 3494-3496.
- GA Kennet et al. SB 242084, a selective and brain penetrant 5-HT2C receptor antagonist. Neuropharmacology 1997, 36(4-5), 609-620.
- GL Dalton et al. Serotonin 1B and 2C receptor interactions in the modulation of feeding behaviour in the mouse. Psychopharmacol. 2006, 185(1), 45-57.
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