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FSEN1
- Soluble in 0.1N HCl(aq), DMSO and EtOH
- MF: C22H22BrN5OS
- MW: 484.41
Description
FSEN1 is an uncompetitive FSP1 inhibitor that sensitizes cancer cells to ferroptosis with an IC50 value of 313 nM. Moreover, FSEN1 synergizes with GPX4 inhibitors and endoperoxide-based ferroptosis inducers.
More Information
| Parent CAS No. | 862808-01-3 |
|---|---|
| Chemical Name | 3-(4-Bromophenyl)-6-((4-(4-methoxyphenyl)piperazin-1-yl)methyl)thiazolo[2,3-c][1,2,4]triazole |
| MFCD | N.A. |
| Short Description | FSP1 inhibitor |
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