Based on 25 reference(s) in Google Scholar 8 10 25

Axon 3786

CAS [1334493-07-0]

MF C29H27F5N2O6S
MW 626.59

  • Purity: 99%
  • Soluble in DMSO and EtOH



BP-1-102 is an orally bioavailable inhibitor of transcription factor Stat3 with an IC50 value of 6.8 μM. BP-1-102 binds Stat3 with an affinity (KD) of 504 nM, blocks Stat3-phospho-tyrosine (pTyr) peptide interactions and Stat3 activation at 4-6.8 μM, and selectively inhibits growth, survival, migration, and invasion of Stat3-dependent tumor cells.

KEYWORDS: BP-1-102 | Supplier | STAT3 inhibitor | BP 1-102 | BP1-102 | CAS [1334493-07-0] | DNA-RNA | STAT3 | Inhibitor | Transcription Factors | Breast cancer | Lung cancer

Size Unit Price Stock
5 mg €90.00 In Stock
25 mg €300.00 In Stock
Special Offers
Size Unit Price Stock
2 x 5 mg €140.00 In Stock
2 x 25 mg €460.00 In Stock
Need more? Bulk Inquiry

The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

Please wait...