ABT-639

Based on 17 reference(s) in Google Scholar 8 10 17

Axon 3785

CAS [1235560-28-7]

MF C20H20ClF2N3O3S
MW 455.91

  • Purity: 99%
  • Optical purity: Optically pure
  • Soluble in 0.1N HCl(aq) and DMSO
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ABT-639

Description

ABT-639 is a peripherally acting, selective and orally bioavailable T-type Ca2+ channel blocker. ABT-639 blocks recombinant human T-type (Ca(v)3.2) Ca2+ channels in a voltage-dependent fashion (IC50 value of 2 μM) and attenuates LVA currents in rat DRG neurons (IC50 value of 8 μM).

KEYWORDS: ABT-639 | Supplier | Ca channel blocker | ABT639 | ABT 639 | CAS [1235560-28-7] | Calcium | Non Selective | Blocker | Ion Channels | Nociceptive pain | Neuropathic pain

Peripherally acting, selective and orally bioavailable T-type Ca2+ channel blocker

Chemical name

(R)-4-Chloro-2-fluoro-N-(2-fluorophenyl)-5-(octahydropyrrolo[1,2-a]pyrazine-2-carbonyl)benzenesulfonamide

Parent CAS No.

[1235560-28-7]

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5 mg €115.00 In Stock
25 mg €390.00 In Stock
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2 x 5 mg €190.00 In Stock
2 x 25 mg €640.00 In Stock
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The purity of Axon Ligands™ is confirmed by HPLC-MS, 1H-NMR and/or microanalysis. Analytical data are available upon request.

Caution: Axon Ligands™ are not fully tested. They are for research purposes only! Not for human consumption!

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