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AC-5216
- XBD173 - Emapunil
- Soluble in DMSO and EtOH
- MF: C23H23N5O2
- MW: 401.46
Description
AC-5216 is a selective translocator protein (TSPO; MBR) ligand. AC-5216 showed high affinity for MBRs prepared from rat whole brain (Ki value of 0.297 nM), rat glioma cells (IC50 value of 3.04 nM) and human glioma cells (IC50 value of 2.73 nM), but only negligible affinity for the other main receptors including central benzodiazepine receptors.
More Information
| Parent CAS No. | 226954-04-7 |
|---|---|
| Chemical Name | N-Benzyl-N-ethyl-2-(7-methyl-8-oxo-2-phenyl-7H-purin-9(8H)-yl)acetamide |
| SMILES | N1C=C2N(C)C(=O)N(CC(=O)N(CC3C=CC=CC=3)CC)C2=NC=1C1C=CC=CC=1 |
| MFCD | MFCD07772312 |
| InChi | InChI=1S/C23H23N5O2/c1-3-27(15-17-10-6-4-7-11-17)20(29)16-28-22-19(26(2)23(28)30)14-24-21(25-22)18-12-8-5-9-13-18/h4-14H,3,15-16H2,1-2H3 |
| InChiKey | NBMBIEOUVBHEBM-UHFFFAOYSA-N |
| CID | 6433109 |
| Short Description | TSPO ligand |
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